Ulwazi ngeMveliso
Igama:Cabazitaxel
Inombolo yeCAS:183133-96-2
Ifomula yemichiza:C45H57NO14
Iinkcukacha:99%
Umbala:umgubo omhlophe okanye omhlophe
Umthombo:ISemi-synthesized nge-10-DAB
Uhlobo:APIs
Imisebenzi yeCabazitaxel
1. Ukuvinjelwa kwe-microtubule aggregation: I-Cabazitaxel inokubophelela kwiiprotheni ze-microtubule ngaphakathi kweeseli ze-tumor kunye nokuthintela ukuhlanganiswa kwe-microtubule, ngaloo ndlela inqanda ukwahlukana kunye nokukhula kweeseli ze-tumor.
2. Ukukhuthazwa kokuzinza kwe-microtubule: I-Cabazitaxel ayivimbeli kuphela i-microtubule aggregation kodwa ikhuthaza ukuzinza kwe-microtubule, okwenza kube nzima ukuba i-microtubules ihlaziywe kwaye ithintele ngokufanelekileyo ukwahlukana kunye nokukhula kweeseli ze-tumor.
3. Ukunciphisa i-tumor blood vessel density: I-Cabazitaxel inokunciphisa ukuxinana kwemithambo yegazi ye-tumor ngokuthintela ukubonakaliswa kwe-vascular endothelial factor growth factor, ukunciphisa ukunikezelwa kwezondlo kwi-tumor, kunye nokusebenzisa i-anti-tumor effect.
Iinkonzo zethu
1.Iimveliso:Ukubonelela ngomgangatho ophezulu, izicatshulwa zezityalo ezisulungekileyo, imathiriyeli ekrwada yamayeza, kunye nabaphakathi bamayeza.
2.Iinkonzo zobugcisa:Izicatshulwa ezenziwe ngokwezifiso ezineenkcazo ezizodwa ngokweemfuno zabathengi.
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