Umgangatho ophezulu we-cabazitaxel amandla omenzi weCabazitaxel

Inkcazelo emfutshane:

I-Carbataxel yinto yekhemikhali esetyenziselwa ukwenza amachiza okulwa nomhlaza.ICarbataxel ngumgubo omhlophe okanye omhlophe ophantse unganyibiliki emanzini, kodwa unyibilika kwi-ethanol.Indlela yayo yokulwa nomhlaza kunye neempawu zifana ne-docetaxel, kwaye ingeyeklasi ye-anti-microtubule drug.Ngokusebenzisa ukudibanisa kunye ne-tubulin, ukukhuthaza ukuhlanganisana kwayo kwii-microtubules, kwangaxeshanye kunokuthintela ezi ziqokelele i-microtubule disassembly, ezizinzisa ii-microtubules, ngaloo ndlela zithintela i-cell mitosis, kunye nokusebenza kweeseli ze-interphase (interphasecellularfunctions).


Iinkcukacha zeMveliso

Iithegi zeMveliso

Ulwazi ngeMveliso

Igama:Cabazitaxel

Inombolo yeCAS:183133-96-2

Ifomula yemichiza:C45H57NO14

Iinkcukacha:99%

Umbala:umgubo omhlophe okanye omhlophe

Umthombo:ISemi-synthesized nge-10-DAB

Uhlobo:APIs

Indima kunye neenzuzo ze-cabataxel

I-1.i-anti-cancer effect: i-carbamazel inempembelelo enamandla yokuchasana nomhlaza, inokuthintela ngokufanelekileyo ukukhula kunye nokusasazeka kweeseli ze-tumor, ifake i-apoptosis yeseli ye-tumor.Xa kuthelekiswa ne-paclitaxel yendalo, i-carbataxel inomsebenzi ophezulu wokuchasana nomhlaza kunye ne-anti-cancer spectrum.

I-2.ukhuseleko: I-Cabataxel kwindlela yokuyila kunye nokuvelisa, gxininisa ekuphuculeni ukhuseleko lwemveliso kunye nokunyamezela.Ngokuguqula kunye nokuphucula ukwakhiwa kweekhemikhali ze-paclitaxel, iziganeko zemiphumo emibi kunye neempembelelo ezimbi zancitshiswa.

I-3.impawu ze-pharmacokinetic: i-carbamazel ineempawu ezingcono ze-pharmacokinetic, ukwenzela ukuba inokuthi ifakwe ngcono kwaye isasazwe emzimbeni, ukwenzela ukuba kuphuculwe umphumo wonyango.

I-4.ukusebenza: i-carbataxel ingasetyenziselwa ukunyanga iintlobo ezahlukeneyo zomhlaza, kubandakanywa umhlaza wamaphaphu, umhlaza wesifuba, umhlaza we-ovarian, umhlaza wesisu, njl njl. Ukusebenza kwayo kunye nokhuseleko kuye kwaqinisekiswa ngokubanzi kwiklinikhi.

I-5.Inkxaso yezeNzululwazi: I-Cabataxel isekelwe kuphando lwenzululwazi yakutshanje kunye nophuhliso lwezobuchwepheshe, kunye nenkxaso yesayensi ethembekileyo.

Iinkonzo zethu

1.Iimveliso:Ukubonelela ngomgangatho ophezulu, izicatshulwa zezityalo ezisulungekileyo, imathiriyeli ekrwada yamayeza, kunye nabaphakathi bamayeza.

2.Iinkonzo zobugcisa:Izicatshulwa ezenziwe ngokwezifiso ezineenkcazo ezizodwa ngokweemfuno zabathengi.

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